Chemisty and Biological Activity
Chemical Formula
C17H15N5O
Chemical Name
N-[3-(9-cyano-2,6,7-triazabicyclo[4.3.0]nona-2,4,7,9-tetraen-5-yl)phenyl]-N- ethyl-ethanamide
Chemical Structure
Molecular Weight
305.334 g/mol
Physical State
Solid
Melting Point
157-159 oC
Water Solubility
Not Available
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
CYP3A4
Primary Drug Target
Name | Benzodiazepine Receptor | Gene Name | BZRP | Synonyms | Peripheral-type benzodiazepine receptor; PBR; PKBS; Mitochondrial benzodiazepine receptor | General Function | Signal transduction mechanisms | Specific Function | Responsible for the manifestation of peripheral-type benzodiazepine recognition sites and is most likely to comprise binding domains for benzodiazepines and isoquinoline carboxamides. May play a role in the transport of porphyrins and heme |
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