Chemisty and Biological Activity
Chemical Formula
C13H24N4O3S
Chemical Name
1-[(4-morpholin-4-yl-1,2,5-thiadiazol-3-yl)oxy]-3-tert-butylamino-propan-2- ol
Chemical Structure
Molecular Weight
316.421 g/mol
Physical State
Solid
Melting Point
201.5-202.5 oC
Water Solubility
2.74 mg/mL
Isoelectric Point
3.9
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
CYP2D6
Primary Drug Target
| Name | Beta-1 Adrenergic Receptor | | Gene Name | ADRB1 | | Synonyms | Beta-1 adrenergic receptor; Beta-1 adrenoceptor; Beta-1 adrenoreceptor | | General Function | Receptor activity and cell communication | | Specific Function | Beta-adrenergic receptors mediate the catecholamine- induced activation of adenylate cyclase through the action of G proteins. This receptor binds epinephrine and norepinephrine with approximatively equal affinity |
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