Chemisty and Biological Activity
Chemical Formula
C16H13ClN2O2
Chemical Name
10-chloro-4-hydroxy-6-methyl-2-phenyl-3,6-diazabicyclo[5.4.0]undeca- 2,8,10,12-tetraen-5-one
Chemical Structure
Molecular Weight
300.739 g/mol
Physical State
Solid
Melting Point
119-121oC
Water Solubility
164 mg/L
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
CYP2C19
Primary Drug Target
| Name | Benzodiazepine Receptor | | Gene Name | BZRP | | Synonyms | Peripheral-type benzodiazepine receptor; PBR; PKBS; Mitochondrial benzodiazepine receptor | | General Function | Signal transduction mechanisms | | Specific Function | Responsible for the manifestation of peripheral-type benzodiazepine recognition sites and is most likely to comprise binding domains for benzodiazepines and isoquinoline carboxamides. May play a role in the transport of porphyrins and heme |
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