Chemisty and Biological Activity
Chemical Formula
C32H53N2O4+
Chemical Name
[3-hydroxy-10,13-dimethyl-2-morpholin-4-yl-16-(1-prop-2-enyl-2,3,4,5- tetrahydropyrrol-1-yl)-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H- cyclopenta[a]phenanthren-17-yl] acetate
Chemical Structure
Molecular Weight
529.774 g/mol
Physical State
Solid
Melting Point
Not Available
Water Solubility
Complete
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
Not Available
Primary Drug Target
| Name | Neuronal acetylcholine receptor protein, alpha-2 subunit precursor | | Gene Name | CHRNA2 | | Specific Function | After binding acetylcholine, the AChR responds by an extensive change in conformation that affects all subunits and leads to opening of an ion-conducting channel across the plasma membrane |
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