Chemisty and Biological Activity
Chemical Formula
C23H27FN4O2
Chemical Name
4-[2-[4-(6-fluorobenzo[d]isoxazol-3-yl)-1-piperidyl]ethyl]-3-methyl-2,6- diazabicyclo[4.4.0]deca-1,3-dien-5-one
Chemical Structure
img=Risperidone_APRD00187_ZOOM.gif
Molecular Weight
410.485 g/mol
Physical State
Solid
Melting Point
170oC
Water Solubility
2.8mg/L
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
CYP2D6
Primary Drug Target
Name | Histamine H1 receptor | Gene Name | HRH1 | Synonyms | Histamine H1 receptor | Specific Function | In peripheral tissues, the H1 subclass of histamine receptors mediates the contraction of smooth muscles, increase in capillary permeability due to contraction of terminal venules, and catecholamine release from adrenal medulla, as well as mediating neurotransmission in the central nervous system |
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