Chemisty and Biological Activity
Chemical Formula
C17H20N4S
Chemical Name
2-methyl-4-(4-methyl-1-piperazinyl)-10H-thieno[2,3-b][1,5]benzodiazepine
Chemical Structure
Molecular Weight
312.434 g/mol
Physical State
Solid
Melting Point
195oC
Water Solubility
Not Available
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
CYP1A2
Primary Drug Target
Name | Muscarinic acetylcholine receptor M5 | Gene Name | CHRM5 | Synonyms | None | Specific Function | The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. Primary transducing effect is PI turnover |
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