Chemisty and Biological Activity
Chemical Formula
C17H17ClN6O3
Chemical Name
[8-(5-chloropyridin-2-yl)-7-oxo-2,5,8-triazabicyclo[4.3.0]nona-1,3,5-trien- 9-yl] 4-methylpiperazine-1-carboxylate
Chemical Structure
Molecular Weight
388.808 g/mol
Physical State
Solid
Melting Point
Not Available
Water Solubility
very slightly soluble
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
CYP2E1; CYP3A4
Primary Drug Target
Name | Benzodiazepine Receptor | Gene Name | BZRP | Synonyms | Peripheral-type benzodiazepine receptor; PBR; PKBS; Mitochondrial benzodiazepine receptor | General Function | Signal transduction mechanisms | Specific Function | Responsible for the manifestation of peripheral-type benzodiazepine recognition sites and is most likely to comprise binding domains for benzodiazepines and isoquinoline carboxamides. May play a role in the transport of porphyrins and heme |
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