Chemisty and Biological Activity
Chemical Formula
C22H26N2O2S
Chemical Name
3-[(1-methylpyrrolidin-2-yl)methyl]-5-(2-phenylsulfonylethyl)-1H-indole
Chemical Structure
Molecular Weight
382.52 g/mol
Physical State
Solid
Melting Point
Not Available
Water Solubility
Readily soluble as hydrobromide formulation
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
CYP3A4
Primary Drug Target
| Name | 5-hydroxytryptamine 1D receptor | | Gene Name | HTR1D | | Synonyms | 5-HT-1D; Serotonin receptor 1D; 5- HT-1D-alpha | | Specific Function | This is one of the several different receptors for 5- hydroxytryptamine (serotonin), a biogenic hormone that functions as a neurotransmitter, a hormone, and a mitogen. The activity of this receptor is mediated by G proteins that inhibit adenylate cyclase activity |
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