Chemisty and Biological Activity
Chemical Formula
C22H26N2O4S
Chemical Name
[2-(2-dimethylaminoethyl)-5-(4-methoxyphenyl)-3-oxo-6-thia-2- azabicyclo[5.4.0]undeca-7,9,11-trien-4-yl]ethanoate
Chemical Structure
Molecular Weight
414.519 g/mol
Physical State
Solid
Melting Point
231oC
Water Solubility
465 mg/L
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
CYP3A4
Primary Drug Target
| Name | Dihydropyridine calcium channel | | Gene Name | CACNG1 | | Synonyms | Voltage-dependent calcium channel gamma-1 subunit; Dihydropyridine- sensitive L-type, skeletal muscle calcium channel gamma subunit | | Specific Function | This protein is a subunit of the dihydropyridine (DHP) sensitive calcium channel. Plays a role in excitation-contraction coupling. The skeletal muscle DHP-sensitive Ca(2+) channel may function only as a multiple subunit complex |
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