Chemisty and Biological Activity
Chemical Formula
C15H10ClN3O3
Chemical Name
6-(2-chlorophenyl)-9-nitro-2,5-diazabicyclo[5.4.0]undeca-5,8,10,12-tetraen- 3-one
Chemical Structure
Molecular Weight
315.711 g/mol
Physical State
Solid
Melting Point
236.5 - 238.5 oC
Water Solubility
<0.1 mg/mL
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
CYP3A4
Primary Drug Target
| Name | GABA-A Receptor | | Gene Name | GABRA1 | | Synonyms | Gamma-aminobutyric-acid receptor alpha-1 subunit precursor; GABA(A receptor | | Specific Function | GABA, the major inhibitory neurotransmitter in the vertebrate brain, mediates neuronal inhibition by binding to the GABA/benzodiazepine receptor and opening an integral chloride channel |
|
