Chemisty and Biological Activity
Chemical Formula
C24H26N2O4
Chemical Name
1-(9H-carbazol-4-yloxy)-3-[2-(2-methoxyphenoxy)ethylamino]propan-2-ol
Chemical Structure
Molecular Weight
406.474 g/mol
Physical State
Solid
Melting Point
114-115 oC
Water Solubility
Practically insoluble (0.583 mg/L)
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
CYP2C9; CYP2D6
Primary Drug Target
| Name | Alpha-1A Adrenergic Receptor | | Gene Name | ADRA1A | | Synonyms | Alpha-1A adrenergic receptor; Alpha 1A-adrenoceptor; Alpha 1A- adrenoreceptor; Alpha-1C adrenergic receptor; Alpha adrenergic receptor 1c | | Specific Function | This alpha-adrenergic receptor mediates its action by association with G proteins that activate a phosphatidylinositol-calcium second messenger system. Its effect is mediated by G(q) and G(11) proteins. |
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