Chemisty and Biological Activity
Chemical Formula
C8H10N4O2
Chemical Name
1,3,7-trimethyl-3,7-dihydropurine-2,6-dione
Chemical Structure
Molecular Weight
194.191 g/mol
Physical State
Solid
Melting Point
238 oC
Water Solubility
22 mg/ml
Isoelectric Point
10.4
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
CYP1A2
Primary Drug Target
| Name | Adenosine A1 receptor | | Gene Name | ADORA1 | | Specific Function | Receptor for adenosine. The activity of this receptor is mediated by G proteins which inhibit adenylyl cyclase |
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