Chemisty and Biological Activity
Chemical Formula
C53H72N2O12+2
Chemical Name
5-[3-[1-[(3,4-dimethoxyphenyl)methyl]-6,7-dimethoxy-2-methyl-3,4-dihydro-1H- isoquinolin-2-yl]propanoyloxy]pentyl 3-[1-[(3,4-dimethoxyphenyl)methyl]- 6,7-dimethoxy-2-methyl-3,4-dihydro-1H-isoquinolin-2-yl]propanoate
Chemical Structure
Molecular Weight
929.145 g/mol
Physical State
Solid
Melting Point
185-194 oC
Water Solubility
Miscible
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
Not Available
Primary Drug Target
| Name | Neuronal acetylcholine receptor protein, alpha-2 subunit precursor | | Gene Name | CHRNA2 | | Specific Function | After binding acetylcholine, the AChR responds by an extensive change in conformation that affects all subunits and leads to opening of an ion-conducting channel across the plasma membrane |
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