Chemisty and Biological Activity
Chemical Formula
C23H36N6O5S
Chemical Name
1-[5-guanidino-2-[(3-methyl-1,2,3,4-tetrahydroquinolin-8- yl)sulfonylamino]pentanoyl]-4-methyl-piperidine-2-carboxylic acid
Chemical Structure
Molecular Weight
508.635 g/mol
Physical State
Solid
Melting Point
Not Available
Water Solubility
Not Available
Isoelectric Point
Not Available
Organisms Affected
Humans and other mammals
Phase 1 Metabolising Enzyme (1-st Step of Metabolism)
Not Available
Primary Drug Target
Name | Prothrombin | Gene Name | F2 | Synonyms | Prothrombin precursor; EC 3.4.21.5; Coagulation factor II | Specific Function | Thrombin, which cleaves bonds after Arg and Lys, converts fibrinogen to fibrin and activates factors V, VII, VIII, XIII, and, in complex with thrombomodulin, protein C | Reaction | Selective cleavage of Arg-|-Gly bonds in fibrinogen to form fibrin and release fibrinopeptides A and B |
|